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Ultima-Anastro
$54.00
Characteristics
ACTIVE HALF-LIFE
2 days
Classification
Non-steroidal aromatase inhibitor
Dosage
0.5-1 mg/day
ACNE
No
WATER RETENTION
No
HBR
No
HEPATOTOXICITY
No
AROMATIZATION
No
Active Substance
FORM
50 pills x 1 mg
Manufacturer
Description
ULTIMA-ARIMIDEX 1mg - ULTIMA PHARMACEUTICALS
50 tabs x 1 mg
Anastrozole, also known as Arimidex, is a non-steroidal aromatase inhibiting drug developed by Zeneca Pharmaceuticals in 1995 for the treatment of breast cancer in women. It is used to inhibit the synthesis of estrogen, making it effective in preventing estrogen-related side effects in male athletes using anabolic steroids.
Purpose and Effects:
- Breast Cancer Treatment: Anastrozole is primarily used in the treatment of breast cancer after surgery and for metastasis in women by inhibiting estrogen synthesis.
- Bodybuilding Use: In male athletes using anabolic steroids, Anastrozole prevents the conversion of testosterone into estradiol (aromatization), thereby avoiding estrogen-related side effects such as gynecomastia, water retention, and fat accumulation.
Dosage:
- The initial recommended dose of Anastrozole is 0.5 mg per day or every other day, depending on the dose of aromatizing steroids being used in the cycle.
Side Effects:
- Anastrozole may suppress the level of good cholesterol (HDL) but generally has fewer side effects compared to other aromatase inhibitors like letrozole.
- Letrozole, another AI, can cause severe side effects such as erectile dysfunction, joint pain, and bones fragility due to its potent suppression of estradiol.
Comparison with SERMs:
- Anastrozole blocks the production of the aromatase enzyme, thereby preventing estradiol generation at the earliest stages, while selective estrogen receptor modulators (SERMs) like tamoxifen or clomiphene only prevent estradiol from binding to receptors.
- SERMs do not reduce estradiol production in the body, allowing estradiol to still circulate in the bloodstream.
Benefits of Anastrozole:
- Anastrozole acts more smoothly compared to letrozole, allowing for a finer adjustment of hormonal balance without completely suppressing estradiol levels.
- Estradiol is essential for maintaining hormonal balance, participating in physiological processes, and promoting muscle mass and strength gain.
Reviews:
- Anastrozole is well-tolerated and effective in preventing estrogen-related side effects in male athletes using anabolic steroids.
- Its smoother action and fewer side effects make it preferable to other aromatase inhibitors like letrozole.
Precautions:
- Anastrozole dosage should be adjusted based on the dose of aromatizing steroids used in the cycle to prevent estrogen-related side effects while maintaining hormonal balance.
Warnings:
- Anastrozole should be kept out of reach of children and is intended for adult use only.
Customer Reviews
12.12.2022
Jay
Verified Purchase
Good stuff, and Ultima is trustworthy.
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